Enise Ece GÜRDAL

Papers

1. Beyer M, Henninger SJ, Haehnel PS, Mustafa AM, Gurdal E, Schubert B, Christmann M, Sellmer A, Mahboobi S, Drube S, Sippl W, Kindler T, Krämer OH, Identification of a highly efficient dual type I/II FMS-like tyrosine kinase inhibitor that disrupts the growth of leukemic cells. Cell Chemical Biology, 2021; https://doi.org/10.1016/j.chembiol.2021.10.011.
2. Turgutalp B, Uslu M, Helvacioglu Sinem, Charehsaz M, Gurdal EE, Sippl W, Kocabas F, Yarim M, Lead Optimization and Structure-Activity Relationship Studies on Myeloid Ecotropic Viral Integration Site 1 Inhibitor. Journal of Medicinal Chemistry, 2021; 64(19):14448-14464.
3. Koksal M, Dedeoglu-Erdogan A, Bader M, Gurdal EE, Sippl W, Reis R, Ozgurbuz M, Sipahi H, Celik T. Design, synthesis and molecular docking of novel 3,5-disubstituted-1,3,4-oxadiazole derivatives as iNOS inhibitors. Archiv der Pharmazie, 2021; 354, e2000469.
4. Güneş SS, Yeşil C, Gurdal EE, Korkmaz EE, Yarım M, Aydın A, Sipahi H. Primum non nocere: In silico prediction of adverse drug reactions of antidepressant drugs. Computational Toxicology, 2021; 18: 100165.
5. Wurzlbauer A, Rüben K, Gürdal E, Chaikuad A, Knapp S, Sippl W, Becker W, Bracher F. How to separate kinase inhibition from undesired monoamine oxidase α inhibition-the development of the DYRK1A inhibitor AnnH75 from the alkaloid harmine, Molecules, 2020; 25, 5962.
6. Alhusadi NA, Turgutalp B, Deniz I, Turkoz Acar E, Sipahi H, Yarim M, Gurdal EE. Synthesis, antimicrobial, antioxidant and molecular docking studies on novel 6-methoxybenzothiazole-piperazine derivatives with propanamide chain, Current Topics in Medicinal Chemistry, 2020; 20(19): 1729-1737.
7. Ozyazici T, Gurdal EE, Orak D, Sipahi H, Ercetin T, Gulcan HO, Koksal M. Synthesis, anti-inflammatory activity and molecular docking studies of some novel Mannich bases of the 1,3,4-oxadiazole-2(3H)-thione scaffold, Archiv der Pharmazie, 2020; 353(7): e2000061.
8. Bobtaina E, Gurdal EE, Durmaz I, Cetin-Atalay R, Yarim M. Synthesis and cytotoxicity studies on novel piperazinylacetamides, Letters in Drug Design & Discovery, 2019; 16: 45-51.
9. Gurdal EE, Turgutalp B, Gulcan HO, Erçetin T, Sahin MF, Durmaz I, Cetin-Atalay R, Nguyen QD, Sippl W, Yarim M. Synthesis of novel benzothiazole-piperazine derivatives and their biological evaluation as acetylcholinesterase inhibitors and cytotoxic agents, Anti-Cancer Agents in Medicinal Chemistry, 2017; 17: 1837-1845.
10. Charehsaz M, Gurdal EE, Helvacıoğlu S, Yarım M. Toxicological evaluation of benzothiazole derivatives carrying piperazine ring, Marmara Pharmaceutical Journal (Journal of Research in Pharmacy), 2017; 21(2):243-250.
11. Gurdal EE, Yarim M, Comparison of separation performance of polysaccaride-based chiral stationary phases in enantioseparation of 1-(4-chlorobenzhydryl)piperazine benzamide derivatives by HPLC, Journal of Analytical Chemistry, 2017; 72(2): 213-216.
12. Gurdal EE, Durmaz I, Cetin-Atalay R, Yarim M, Cytotoxic activities of some benzothiazole-piperazine derivatives, Journal of Enzyme Inhibition & Medicinal Chemistry, 2015; 30(4): 649-654.
13. Gurdal EE, Buclulgan E, Durmaz I, Cetin-Atalay R, Yarim M, Synthesis and anticancer activity evaluation of some benzothiazole-piperazine derivatives, Anti-Cancer Agents in Medicinal Chemistry, 2015; 15: 382-389.
14. Gurdal EE, Durmaz I, Cetin-Atalay R, Yarim M, Synthesis and cytotoxicity studies of novel benzhydrylpiperazine carboxamide and thioamide derivatives, Journal of Enzyme Inhibition & Medicinal Chemistry, 2014; 29(2): 205-214.
15. Gurdal EE, Yarim M, Durmaz I, Cetin-Atalay R, Cytotoxic activities of some novel benzhydrylpiperazine derivatives, Drug Research, 2013; 63(3): 121-128.
16. Us D, Berk B, Gurdal E, Aytekin N, Kocagoz T, Caglayan B, Kurnaz IA, Erol DD, Mannich base derivatives of 3-hydroxy-6-methyl-4h-pyran-4-one with antimicrobial activity, Turkish Journal of Chemistry, 2010; 34: 447-456.
17. Us D, Gurdal E, Berk B, Öktem S, Kocagoz T, Caglayan B, Kurnaz IA, Erol DD, 4H-Pyran-4-one derivatives: Leading molecule for preparation of compounds with antimycobacterial potential, Turkish Journal of Chemistry, 2009; 33: 803-812.